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KROMOZOME

API Portfolio

Oncology APIs

Product Therapeutic Use Regulatory / Grade
Axitinib Anti-Cancer / TKI USDMF
Azacitidine Anti-Cancer USDMF
Bendamustine HCl Monohydrate Anti-Cancer USDMF
Bicalutamide Anti-Cancer USDMF
Bortezomib Anti-Cancer IP / USDMF
Busulfan Anti-Cancer CEP, USDMF
Cabazitaxel Anti-Cancer USDMF
Calcium Folinate Anti-Cancer (adjunct) USP/BP/EP/IP
Capecitabine Anti-Cancer CEP, USDMF
Carboplatin Anti-Cancer USP/Ph.Eur/BP
Carmustine Anti-Cancer USP/Ph.Eur/BP
Chlorambucil Anti-Cancer USP/BP/EP/IP
Cisplatin Anti-Cancer USP/Ph.Eur/BP/IP
Clofarabine Anti-Cancer USDMF
Crizotinib Anti-Cancer In-house
Cyclophosphamide Anti-Cancer USDMF, CEP
Fulvestrant Anti-Cancer USP/IP
Gemcitabine HCl Anti-Cancer CEP, USDMF
5-Fluorouracil Anti-Cancer USP/BP/EP/IP
Ibrutinib Anti-Cancer / BTK inhibitor USDMF
Imatinib Mesylate Anti-Cancer CEP, USDMF
Irinotecan HCl Trihydrate Anti-Cancer CEP, USDMF
Lenalidomide Anti-Cancer USDMF
Lenvatinib Mesylate Anti-Cancer USDMF
Melphalan / Melphalan HCl Anti-Cancer IP/USP, USDMF
Methotrexate Anti-Cancer USP/Ph.Eur/BP/IP
Mitomycin Anti-Cancer USP/BP/EP/IP
Nilutamide Anti-Cancer Ph.Eur
Oxaliplatin Anti-Cancer USP/Ph.Eur/BP
Paclitaxel Anti-Cancer USP/Ph.Eur/BP/IP
Palbociclib (N-1/N-2) Anti-Cancer Advanced Intermediate
Pemetrexed Disodium Anti-Cancer USP, USDMF
Zoledronic Acid Anti-Cancer / Bone IP, USDMF
Cytarabine Anti-Cancer USP/Ph.Eur/BP/IP
Dasatinib (incl. Monohydrate) Anti-Cancer DMF Available / In-house
Decitabine Anti-Cancer USDMF
Docetaxel Trihydrate Anti-Cancer USP/Ph.Eur/IP/BP
Enzalutamide Anti-Cancer USDMF
Erlotinib HCl Anti-Cancer USDMF
Etoposide Anti-Cancer USP/Ph.Eur/BP/IP
Fludarabine Phosphate Anti-Cancer Ph.Eur/In-house
Pomalidomide Anti-Cancer USDMF
Sunitinib Malate Anti-Cancer USDMF
Temozolomide Anti-Cancer USP/IP, CEP, USDMF
Thalidomide Anti-Cancer USDMF
Trofosfamide Anti-Cancer In-house
Vinblastine Sulphate Anti-Cancer USP/Ph.Eur/BP/IP
Vincristine Sulphate Anti-Cancer USP/Ph.Eur/IP
Vinorelbine Tartrate Anti-Cancer USP/Ph.Eur/BP/IP
Zoledronic Acid Anti-Cancer / Bone IP, USDMF
Cytarabine Anti-Cancer USP/Ph.Eur/BP/IP
Dasatinib (incl. Monohydrate) Anti-Cancer DMF Available / In-house
Decitabine Anti-Cancer USDMF
Docetaxel Trihydrate Anti-Cancer USP/Ph.Eur/IP/BP
Enzalutamide Anti-Cancer USDMF
Erlotinib HCl Anti-Cancer USDMF
Etoposide Anti-Cancer USP/Ph.Eur/BP/IP
Fludarabine Phosphate Anti-Cancer Ph.Eur/In-house
Pomalidomide Anti-Cancer USDMF
Sunitinib Malate Anti-Cancer USDMF
Temozolomide Anti-Cancer USP/IP, CEP, USDMF
Thalidomide Anti-Cancer USDMF
Trofosfamide Anti-Cancer In-house
Vinblastine Sulphate Anti-Cancer USP/Ph.Eur/BP/IP
Vincristine Sulphate Anti-Cancer USP/Ph.Eur/IP
Vinorelbine Tartrate Anti-Cancer USP/Ph.Eur/BP/IP

Oncology Intermediates (N-1 / N-2)

Specialised in advanced N-1 / N-2 oncology intermediate chemistry — developed and supplied at commercial scale.

Product Therapeutic Use CAS No.
6,7-Dimethoxy-4-chloroquinoline Cabozantinib / Tivozanib 35654-56-9
2-Amino-N-(2-chloro-6-methylphenyl)-5-thiazolecarboxamide Dasatinib (N-2) 302964-24-5
N-(2-Chloro-6-methylphenyl)-2-[(6-chloro-2-methyl-4-pyrimidinyl)amino]-5-thiazolecarboxamide Dasatinib (N-1) 302964-08-5
3-Aminophenylacetylene Erlotinib side chain 54060-30-9
6,7-Bis-(2-methoxyethoxy)-4(3H)-quinazolinone Erlotinib (N-2) 179688-29-0
R-3-(4-Phenoxy-phenyl)-1-piperidin-3-yl-1H-pyrazolo[3,4-d]pyrimidin-4-amine Ibrutinib (N-1) 1022150-12-4
3-(4-Phenoxy Phenyl)-1H-pyrazole[3,4-d]pyrimidin-4-Amine Ibrutinib (N-2) 330786-24-8
Methyl-(S)-N-Ethoxycarbonyl-4-Amino phenylalaninate Melphalan (N-1) 169472-17-7
4-Amino-L-phenyl-N-phthalylalanine ethyl ester Melphalan (N-2) 74743-23-0
N-(2-chloropyrimidin-4-yl)-N,2,3-trimethylindazol-6-amine Pazopanib (N-1) 444731-75-3
5-Amino-2-methyl-benzenesulfonamide Pazopanib side chain 6973-07-9
4-[2-(2-Amino-4,7-dihydro-4-oxo-1H-pyrrolo[2,3-d]pyrimidin-5-yl)ethyl]benzoic acid Pemetrexed (N-2) 137281-39-1
4-(4-Aminophenoxy)-N-methylpyridine-2-carboxamide Sorafenib (N-2) 284462-37-9
Methyl-4-(4-aminophenyl)butyrate Chlorambucil (N-2) 20637-09-6
Methyl-4-{4-[Bis(2-Hydroxyethyl)Amino]Phenyl}Butanoate Chlorambucil (N-1) 130198-76-4
3-(4-methyl-1H-imidazol-1-yl)-5-(trifluoromethyl)aniline Nilotinib (N-1) 641571-11-1
6-Bromo-2-chloro-8-cyclopentyl-5-methylpyrido[2,3-d]pyrimidin-7(8H)-one Palbociclib (N-1) 1016636-76-2
tert-Butyl 4-(6-aminopyridin-3-yl)piperazine-1-carboxylate Palbociclib (N-2) 571188-59-5
Beta-D-Ribofuranose 1,2,3,5-tetraacetate Azacitidine (N-1) 13035-61-5
5-Azacytosine Azacitidine (N-2) 931-86-2
1,2,3-Triacetyl-5-deoxy-D-ribose Capecitabine (N-1) 62211-93-2
4-Chloro-7H-pyrrolo[2,3-d]pyrimidine Ruxolitinib (N-1) 3680-69-1
4-(4,5-Dihydro-1H-pyrazol-4-yl)-7-((2-(trimethylsilyl)ethoxy)methyl)-7H-pyrrolo[2,3-d]pyrimidine Ruxolitinib (N-2) 941685-27-4
N-(4-cyano-3-(trifluoromethyl)phenyl)-2-methyloxirane-2-carboxamide Bicalutamide (N-1) 90357-51-0
N-[3-Chloro-4-(3-fluorobenzyloxy)phenyl]-6-iodoquinazolin-4-amine Lapatinib (N-1) 231278-20-9
5-[Bis(2-hydroxyethyl)amino]-1-methyl-1H-benzimidazole-2-butanoic acid ethyl ester Bendamustine (N-1) 3543-74-6
1-Methyl-5-amino-1H-benzimidazole-2-butanoic acid ethyl ester Bendamustine (N-2) 3543-73-5
2,6-Dioxopiperidine-3-ammonium chloride Thalidomide / Pomalidomide / Lenalidomide (N-2) 24666-56-6
Methyl 2-bromomethyl-3-nitrobenzoate Lenalidomide (N-2) 98475-07-1
4-Methyl-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]benzoic acid Nilotinib (N-2) 641569-94-0

Cardiovascular & Metabolic APIs

Product Therapeutic Use Regulatory / Grade
Amlodipine Besilate Anti-Hypertensive Multi-market DMF/CEP
Alfuzosin HCl Anti-Hypertensive / BPH EU CEP, US DMF
Atorvastatin Calcium Anti-Hyperlipidemic IP/USP/Ph.Eur
Bempedoic Acid Anti-Hyperlipidemic In-house
Bisoprolol Fumarate Beta Blocker Multi-market DMF/CEP
Bumetanide Diuretic EU CEP
Carvedilol Beta Blocker 72956-09-3
Clonidine HCl Anti-Hypertensive EU CEP, US DMF
Doxazosin Mesylate Anti-Hypertensive / BPH US DMF
Ezetimibe Anti-Hyperlipidemic / Cardiovascular 163222-33-1
Finerenone Chronic Kidney Disease 1050477-31-0
Hydrochlorothiazide Diuretic Multi-market DMF/CEP
Irbesartan Anti-Hypertensive (ARB) IP/EP/USP
Labetalol HCl Anti-Hypertensive US DMF
Macitentan Pulmonary Hypertension In-house
Valsartan Anti-Hypertensive (ARB) IP/USP/Ph.Eur
Calcium Dobesilate Monohydrate Vasoprotective CEP 2023-106
Diosmin Hesperidin Vasoprotective US DMF
Rizatriptan Benzoate Anti-Migraine EU CEP
Prasugrel Anti-Platelet US DMF
Nebivolol Hydrochloride Beta Blocker US DMF
Ranolazine Anti-Anginal US DMF
Resmetirom Liver Disorders (MASH) 920509-32-6
Rivaroxaban Anti-Coagulant EU CEP, US DMF
Apixaban Anti-Coagulant EU/EDMF, US DMF
Sacubitril Sodium Hypertension / Heart Failure US DMF
Sacubitril Valsartan Hypertension / Heart Failure US DMF
Simvastatin Anti-Hyperlipidemic In-house
Tadalafil Cardiovascular / Urology EU CEP, US DMF

CNS, Neurology & Anesthetic APIs

Product Therapeutic Use Regulatory / Grade
Lacosamide Anti-Convulsant US DMF
Lamotrigine Anti-Convulsant EU CEP, US DMF
Brivaracetam Anti-Convulsant In-house
Cenobamate Anti-Convulsant US DMF
Carbamazepine Anti-Convulsant IP/BP/EP/USP
Oxcarbazepine Anti-Convulsant CEP 2021-340
Phenytoin Sodium Anti-Convulsant US DMF
Tizanidine HCl Muscle Relaxant / CNS EU CEP, US DMF
Quetiapine Fumarate Anti-Psychotic In-house / IP/USP
Lurasidone HCl Anti-Psychotic US DMF
Brexpiprazole Atypical Anti-Psychotic US DMF
Vortioxetine HBr Anti-Depressant US DMF
Suvorexant Hypnotic In-house
Lemborexant Hypnotic 1369764-02-2
Trazodone HCl Anti-Depressant CEP-2023-228, US DMF
Citicoline Sodium Neuro-Protective US DMF
Lumateperone Tosylate Anti-Psychotic 1187020-80-9
Rimegepant Anti-Migraine 1289023-67-1
Pimavanserin Anti-Psychotic (Parkinson's) US DMF
Guanfacine CNS / ADHD US DMF
Topiramate Anti-Convulsant / Migraine US DMF
Rocuronium Bromide Muscle Relaxant 119302-91-9
Etomidate Anesthetic In-house
Propofol Anesthetic In-house
Prilocaine Anesthetic IP/BP/EP/USP

Anti-Infective APIs

Product Therapeutic Use Regulatory / Grade
Acyclovir Anti-Viral IP/BP/EP/USP
Valacyclovir HCl Anti-Viral In-house
Valganciclovir Anti-Viral In-house
Famciclovir Anti-Viral US DMF, TGA
Penciclovir Anti-Viral In-house
Oseltamivir / Oseltamivir Phosphate Anti-Viral IP/EP
Baloxavir Marboxil Anti-Viral 1985606-14-1
Entecavir Monohydrate Hepatitis B USP/IP/Ph.Eur
Sofosbuvir Hepatitis C In-house
Daclatasvir Dihydrochloride Hepatitis C 1009119-65-6
Ritonavir Anti-Viral IP/USP/Ph.Eur
Amantadine Hydrochloride Anti-Viral US DMF
Fluconazole Anti-Fungal USP/IP/EP/JP
Miconazole Nitrate Anti-Fungal IP/USP/EP/JP
Tavaborole Anti-Fungal 174671-46-6
Clotrimazole Anti-Fungal In-house
Econazole Nitrate Anti-Fungal In-house
Fosfomycin Calcium / Sodium / Trometamol Urinary Tract Infection US DMF
Amoxicillin Trihydrate Antibiotic In-house
Ampicillin Trihydrate Antibiotic In-house
Cloxacillin Sodium Antibiotic In-house
Bedaquiline Fumarate Anti-Tuberculosis 845533-86-0
Pretomanid Anti-Tuberculosis 187235-37-6
Aminosalicylate Sodium Anti-Tuberculosis 6018-19-5
Amino Salicylic Acid Anti-Bacterial / Anti-TB 65-49-6
Ethopabate Anti-Coccidial (Veterinary) 59-06-3
Chlorhexidine (Base / Diacetate / Digluconate / Dihydrochloride) Disinfectant US DMF, CEP
Octenidine Dihydrochloride Disinfectant DMF, KFDA, ASMF
Polyhexamethylene Biguanide (PHMB) Disinfectant US DMF
L-Carbocisteine Mucolytic / Anti-Bacterial 638-23-3
Metronidazole Antibiotic EU CEP, US DMF
Metronidazole Benzoate Antibiotic CEP 2023-417
Norfloxacin Antibiotic IP/BP/EP/USP
Ofloxacin Antibiotic IP/BP/EP/USP
Linezolid Antibiotic In-house
Tedizolid Phosphate Antibiotic 856867-55-5

Respiratory & Anti-Allergic APIs

Product Therapeutic Use Regulatory / Grade
Formoterol Fumarate Anti-Asthmatic In-house
Arformoterol Tartrate Anti-Asthmatic In-house
Doxofylline Anti-Asthmatic US DMF, KFDA
Montelukast Sodium Anti-Asthmatic US DMF
Cetirizine Dihydrochloride Anti-Allergic In-house
Chlorpheniramine Maleate Anti-Allergic In-house
Pheniramine Maleate Anti-Allergic In-house
Fexofenadine HCl Anti-Allergic In-house
Bilastine Anti-Histamine 202189-78-4
Ambroxol HCl Mucolytic / Expectorant EU CEP
Noscapine Anti-Tussive US DMF
Dimenhydrinate Anti-Emetic / Anti-Vertigo In-house
Diphenhydramine HCl Anti-Histamine In-house
Cetylpyridinium Chloride Antiseptic (throat/oral) In-house

Gastro, Urology & Other Specialty APIs

Product Therapeutic Use Regulatory / Grade
Rabeprazole Sodium Gastro (PPI) IP/USP
Elobixibat GI & IBS 439087-18-0
Vonoprazan Fumarate Gastro (PCAB) 881681-01-2
Mesalamine Anti-Inflammatory (IBD) In-house
Famotidine Anti-Ulcer In-house
Metoclopramide HCl Anti-Emetic 54143-57-6
Carglumic Acid Hyperammonaemia 1188-38-1
Tamsulosin HCl UTI / BPH IP/EP/USP/BP
Silodosin Hypertension / BPH 160970-54-7
Vibegron Overactive Bladder 1190389-15-1
Etoricoxib NSAID / Anti-Inflammatory 202409-33-4
Meloxicam NSAID In-house
Piroxicam NSAID In-house
Bromfenac Sodium NSAID In-house
Polmacoxib NSAID In-house
Loxoprofen Sodium NSAID 80382-23-6
Mefenamic Acid NSAID In-house
Papaverine HCl Vasodilator US DMF
Varenicline Tartrate Smoking Cessation US DMF
Febuxostat Anti-Gout In-house
Diacerein Anti-Osteoarthritic In-house
Ketoprofen / Dexketoprofen Trometamol Analgesic In-house
Olmesartan Medoxomil Anti-Hypertensive In-house
Fenspiverinium Bromide Antispasmodic In-house
Pitofenone HCl Antispasmodic In-house
Deferasirox Iron Chelator US DMF, EU CEP
Ferric Carboxymaltose Iron Replacement Agent DMF, KFDA
Ferrous Ascorbate Anti-Anemic In-house
Amisulpride Anti-Psychotic 71675-85-9
Oxymetazoline HCl / Xylometazoline HCl Decongestant IP/BP/EP/USP
Terbutaline Sulphate Broncho-dilator In-house
Isoxsuprine HCl Vasodilator In-house